An improved method for the palladium-catalyzed amination of aryl iodides.

نویسندگان

  • M H Ali
  • S L Buchwald
چکیده

Aryl iodides are coupled with amines to give the corresponding arylamines in high yield in the presence of palladium, a suitable ligand, and NaOt-Bu. Functionalized aryl iodides give good yields of the corresponding arylamines when Cs(2)CO(3) is substituted as the base.

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عنوان ژورنال:
  • The Journal of organic chemistry

دوره 66 8  شماره 

صفحات  -

تاریخ انتشار 2001